Minofu Supplement Anti Estrogen Steroids White Powder Tamoxifen Citrate Nolvadex
Tsatanetsatane Wachangu
Mankhwala: Nolvadex (Tamoxifen Citrate)
Nambala ya CAS: 54965-24-1
MF: C26H29NO
MW: 371.51
Chiyero: 99%
Malo otentha: 482.3°C pa 760 mmHg
Kusungirako: Kusindikizidwa mu 2 ºC -8 ºC
Malo osungunuka: 140-144 °C
kung'anima: 356.5ºC
Kapangidwe:
Einecs No: 234-118-0
Standard: Enterprise Standard
Mankhwala Ena Oletsa Khansa: Tamoxifen Citrate, Clomiphene Citrate, Toremifene Citrate, Anastrozole, Raloxifene hydrochloride, Fulvestrant, Letrozole, Crotamiton
Kagwiritsidwe:Tamoxifen ndi mahomoni achikazi omwe amatha kuletsa zochita za estrogen, nthawi zambiri amagwiritsidwa ntchito pochiza mitundu ina ya khansa ya m'mawere mwa amuna ndi akazi.
Chithandizo cha Khansa Steroids timapereka
Tamoxifen Citrate | non-steroidal wothandizira |
Exemestane | Aromatase inhibitor |
Anastrozole | amagwiritsidwa ntchito pogwiritsira ntchito ma steroid ochuluka kwambiri |
Stanozolol | Kudula Zozungulira |
Toremifene Citrate | non-steroidal selective Estrogen receptor modulator |
Drostanolone Propionate | Anabolic Steroid |
Methenolone Enanthate | mapuloteni timadzi kutengera mphamvu ya chiwindi |
17-methyltestosterone | androgen ndi Albumen Assimilation steroids |
Fluoxymesterone | angagwiritsidwe ntchito ngati mankhwala mankhwala |
Formestan | Amagwiritsidwa ntchito ngati choletsa ma enzyme |
Chinsinsi cha Nolvadex
Ufa: pa 1 gramu ya Tamoxifen Citrate
Amapanga: ndende yapamwamba kwambiri - 20 mg/ml
Zofunikira:
1 gramu ya Tamoxifen citrate
1 beaker yoyenera kusunga kuchuluka kwa zakumwa
19.6 ml ya glycerol
29.4 ml ya 190 Umboni wa Mbewu Mowa
Ufa: pa 1 gramu ya Tamoxifen Citrate
Amapanga: ndende yapamwamba kwambiri - 20 mg/ml
Zofunikira:
1 gramu ya Tamoxifen citrate
1 beaker yoyenera kusunga kuchuluka kwa zakumwa
9.8 ml ya PEG 600
39.2 ml ya 190 Umboni Wambewu Mowa
Kugwiritsa ntchito kwa Nolvadex ndi mlingo
Khansa ya M'mawere | 10 mpaka 20 mg pakamwa kawiri pa tsiku |
Kwa khansa ya m'mawere ya metastatic | 20 mpaka 40 mg amaperekedwa mogawanika |
Amayi omwe ali ndi Ductal Carcinoma | 20 mg tsiku lililonse kwa zaka 5 |
Chepetsani kuchuluka kwa khansa ya m'mawere | 20 mg tsiku lililonse kwa zaka 5 |
Node-positive khansa ya m'mawere, axillary dissection | 10 mg pakamwa 2 mpaka 3 pa tsiku kwa zaka 5. |
Atsikana azaka zapakati pa 2 mpaka 10 ndi McCune-Albright Syndrome | 20 mg tsiku lililonse kwa chaka chimodzi |
Ntchito ya Nolvadex
1: Tamoxifen Citrate Gwiritsani ntchito Cancer
Tamoxifen citrate | Zavomerezedwa kupewa: Khansa ya m'mawere mwa amayi omwe ali pachiwopsezo chachikulu cha matendawa. |
Khansara ya m'mawere mwa amayi ndi abambo | |
akuphunziridwa pochiza mitundu ina ya khansa. |
2: Ubwino wa Tamoxifen
A. Tamoxifen imachepetsa kapena kuletsa kukula kwa maselo a khansa omwe alipo kale m'thupi.Imathandiza kuti khansa ya m'mawere yoyambirira isabwerere ndipo imathandizira kupewa khansa yatsopano m'mawere ena.Zimachepetsanso chiopsezo cha khansa ya m'mawere mwa amayi omwe ali ndi chiopsezo chachikulu cha matendawa.
B. Tamoxifen amagwiritsidwa ntchito pofuna kupewa ndi kuchiza khansa ya m'mawere yomwe imayesa zabwino za estrogen receptors (ER +).Imatsekereza zotsatira zomwe timadzi ta estrogen timakhala ndi ma cell a khansa ndikuchepetsa mwayi woti khansa ya m'mawere ikule.Nthawi zambiri amatchedwa "anti-estrogen."
C. Tamoxifen imathandiza kwambiri kuchepetsa chiopsezo cha khansa ya m'mawere.Kwa amayi omwe ali ndi khansa ya m'mawere, tamoxifen imachepetsanso chiopsezo cha khansa ya m'mawere kumbali ina (contralateral)
D. Kwa amayi omwe ali ndi postmenopausal, chithandizo chamagulu awiri pogwiritsa ntchito tamoxifen ndiyeno aromatase inhibitor, monga anastrozole (Arimidex), exemestane (Aromasin), kapena letrozole (Femara) angagwire ntchito bwino kusiyana ndi kumwa tamoxifen kokha.